Synthesis and Structure−Activity Relationship Studies of N‐Benzyl-2- phenylpyrimidin-4-amine Derivatives as Potent USP1/UAF1 Deubiquitinase Inhibitors with Anticancer Activity against Nonsmall Cell…

By T. Dexheimer, Andrew S. Rosenthal, D. Luci, Qin Liang, M. Villamil, Junjun Chen, Hongmao Sun, Edward H. Kerns, Anton Simeonov, A. Jadhav and 2 more. 2014

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1. J. Harrigan
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4. Stephen P. Jackson
5. Yosef Shiloh

Citations in the corpus

• Deubiquitylating enzymes and drug discovery: emerging opportunities (2017, background): “So far, however, little progress has been made in advancing selective USP1 inhibitors into clinical development.”